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Kinase

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Items 1 to 30 of 45 total

  1. A83-01, TGF-β Inhibitor

    $59.00
    Catalog No. M60021
    A potent and selective TGF-β pathway inhibitor (targeting ALK4, ALK5 and ALK7).
  2. AA92593, Antagonist of Melanopsin-mediated Photo-transduction

    $139.00
    Catalog No. M60143
    A potent and selective small molecule antagonist of melanopsin-mediated photo-transduction.
  3. AZD6244 (Selumetinib), MEK Inhibitor

    $109.00
    Catalog No. M60067
    A potent and highly selective non-ATP competitive MEK inhibitor in clinical trials.
  4. BI-2536, PLK1 and BRD4 Dual Inhibitor

    $119.00
    Catalog No. M60171
    BI-2536 is a potent inhibitor of PLK1 (Polo-like kinase 1) and BRD4 in clinical trials.
  5. BIBW2992(Afatinib), EGFR Inhibitor

    $109.00
    Catalog No. M60065-5s
    A potent and selective irreversible inhibitor of EGFR/HER2 in clinical trials.
  6. CP-690550, JAK Inhibitor

    $79.00
    Catalog No. M60033
    A potent and selective pan-JAK Inhibitor in clinical trials for rheumatoid arthritis.
  7. CUDC-101, HDAC/EGFR/HER2 Inhibitor

    $69.00
    Catalog No. M60092
    A potent multi-target inhibitor targeting HDAC, EGFR and HER2 in clinical trial.
  8. CX-4945, CK2 (Casein Kinase 2) Inhibitor

    $129.00
    Catalog No. M60267
    A potent, selective and bioavailable CK2 (Casein Kinase 2) Inhibitor.
  9. DASA-58 (ML203), Pyruvate Kinase M2 (PKM2) Activator

    $109.00
    Catalog No. M60305
    A potent and selective Pyruvate kinase M2 (PKM2) activator.
  10. GDC-0349, mTOR Inhibitor

    $129.00
    Catalog No. M60110
    A potent and selective ATP-competitive inhibitor of mTOR in clinical trials.
  11. GDC-0449 (Vismodegib), Hedgehog Antagonist

    $79.00
    Catalog No. M60034
    A potent and specific hedgehog pathway inhibitor approved by FDA
  12. GDC-0941, PI3K Inhibitor

    $79.00
    Catalog No. M60111
    A highly potent, selective and orally bioavailable class-I PI3K kinase inhibitor.
  13. GNF4877, β Cell Proliferation Inducer

    $159.00
    Catalog No. M60294
    A highly potent and selective small molecule that promotes pancreatic β cell proliferation in rodent and human primary islets.
  14. GNF7156, β Cell Proliferation Inducer

    $139.00
    Catalog No. M60293
    A highly potent and selective small molecule that promotes pancreatic β cell proliferation in rodent and human primary islets.
  15. Go6893, PKC Inhibitor

    $129.00
    Catalog No. M60273
    A potent pan-PKC inhibitor.
  16. Harmine, DYRK1A Inhibitor

    $29.00
    Catalog No. M60241
    A potent, selective and orally bioavailable DYRK1A inhibitor.
  17. HG-10-102-01, LRRK2 Inhibitor

    $139.00
    Catalog No. M60061
    A brain penetrant potent and selective inhibitor of wild-type LRRK2 and the G2019S mutant.
  18. ID-8, DYRK Inhibitor

    $89.00
    Catalog No. M60102
    A potent and selective small molecule inhibitor of dual-specificity tyrosine phosphorylation- regulated kinase (DYRK).
  19. INDY, DYRK1A/B Inhibitor

    $79.00
    Catalog No. M60242
    A potent and selective DYRK1A/B inhibitor.
  20. IRE-3, IRE1a Modulator

    $129.00
    Catalog No. M60167
    A highly potent and selective small molecule modulator of IRE1α.
  21. LDN-193189, BMP inhibitor

    $79.00
    Catalog No. M60008
    A highly potent and selective BMP pathway inhibitor (selective for ALK2 and ALK3); can replace Noggin protein in cellular and in vivo use.
  22. LY2109761, TGFβ Inhibitor

    $109.00
    Catalog No. M60035
    A novel potent and selective TGFβ receptor type I and type II (TβRI/II) dual inhibitor with Ki of 38 nM and 300 nM respectively.
  23. LY2157299, TGFβ Inhibitor

    $169.00
    Catalog No. M60064
    A novel potent and selective TGFβ receptor type I and type II (TβRI/II) inhibitor with IC50 of 86 nM and 2 nM respectively.
  24. LY2784544, JAK2 inhibitor

    $129.00
    Catalog No. M60079
    A highly potent and selective mutant JAK2 (V617F) inhibitor.
  25. LY294002, PI3K/BET Dual Inhibitor

    $79.00
    Catalog No. M60157
    A potent and selective small molecule PI3K and BET bromodomain dual inhibitor.
  26. MEK162 (ARRY-162), MEK Inhibitor

    $119.00
    Catalog No. M60080
    A highly potent, selective, and orally bioavailable MEK inhibitor in clinical trials.
  27. MLN8237 (Alisertib), Aurora A inhibitor

    $119.00
    Catalog No. M60093
    A highly potent and selective Aurora A inhibitor with >200-fold selective towards Aurora B.
  28. MRT68921, Autophagy Kinase ULK1/2 Inhibitor

    $109.00
    Catalog No. M60311
    A potent, selective and dual autophagy kinase ULK1/2 inhibitor.
  29. NVP-BGT226, PI3K/mTOR Dual Inhibitor

    $89.00
    Catalog No. M66050
    A PI3K/mTOR dual inhibitor in clinical trials for advanced solid tumors.
  30. NVP-BKM120, PI3K Inhibitor BKM120

    $89.00
    Catalog No. M66051
    A selective PI3K Inhibitor in clinical trials for advanced solid tumors.
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