Description
ZEN-3411 is a BET inhibitor with IC50s of 0.05, 0.05 and 0.06 μM for BRD4(BD1), BRD4(BD2) and BRD4(BD1BD2), respectively. ZEN-3411 can be used to form PROTACs to induce degradation of BRD4.
Product information
CAS Number: 1952264-36-6
Molecular Weight: 360.41
Formula: C21H20N4O2
Chemical Name: 6-(3,5-dimethyl-1,2-oxazol-4-yl)-1-{[4-(oxiran-2-yl)phenyl]methyl}-1H-1,3-benzodiazol-4-amine
Smiles: CC1ON=C(C)C=1C1C=C(N)C2N=CN(CC3C=CC(=CC=3)C3CO3)C=2C=1
InChiKey: XINQCOMOQIYWTG-UHFFFAOYSA-N
InChi: InChI=1S/C21H20N4O2/c1-12-20(13(2)27-24-12)16-7-17(22)21-18(8-16)25(11-23-21)9-14-3-5-15(6-4-14)19-10-26-19/h3-8,11,19H,9-10,22H2,1-2H3
Technical Data
Appearance: Solid Power
Purity: ≥98% (or refer to the Certificate of Analysis)
Shipping Condition: Shipped under ambient temperature as non-hazardous chemical or refer to Certificate of Analysis
Storage Condition: Dry, dark and -20 oC for 1 year or refer to the Certificate of Analysis.
Shelf Life: ≥12 months if stored properly.
Stock Solution Storage: 0 - 4 oC for 1 month or refer to the Certificate of Analysis.
Drug Formulation: To be determined
HS Tariff Code: 382200
Products are for research use only. Not for human use.
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