[Orn5]-URP


Catalog No. Size PriceQuantity
M21964-C Contact sales@xcessbio.com for quotation $100Unavailable

Description

[Orn5]-URP is a potent and selective pure antagonist of Urotensin-II receptor (UT), with an pEC50 of 7.24. [Orn5]-URP displays no agonist activity.

Product information

CAS Number: 782485-03-4

Molecular Weight: 1003.20

Formula: C48H62N10O10S2

Chemical Name: (2S)-2-[(Z)-{[(4R,7S,10S,13S,16S,19R)-19-[(Z)-[(2R)-2-amino-1-hydroxypropylidene]amino]-10-(3-aminopropyl)-16-benzyl-6,9,12,15,18-pentahydroxy-7-[(4-hydroxyphenyl)methyl]-13-[(1H-indol-3-yl)methyl]-1,2-dithia-5,8,11,14,17-pentaazacycloicosa-5,8,11,14,17-pentaen-4-yl](hydroxy)methylidene}amino]-3-methylbutanoic acid

Smiles: CC(C)[C@H](/N=C(\O)/[C@@H]1CSSC[C@H](/N=C(\O)/[C@@H](C)N)C(O)=N[C@@H](CC2C=CC=CC=2)C(O)=N[C@@H](CC2=CNC3=CC=CC=C23)C(O)=N[C@@H](CCCN)C(O)=N[C@@H](CC2C=CC(O)=CC=2)C(O)=N1)C(O)=O |t:20,32,48,56,69|

InChiKey: BPLKRLYKWHXTMO-JKFZISEOSA-N

InChi: InChI=1S/C48H62N10O10S2/c1-26(2)40(48(67)68)58-47(66)39-25-70-69-24-38(56-41(60)27(3)50)46(65)54-35(20-28-10-5-4-6-11-28)43(62)55-37(22-30-23-51-33-13-8-7-12-32(30)33)45(64)52-34(14-9-19-49)42(61)53-36(44(63)57-39)21-29-15-17-31(59)18-16-29/h4-8,10-13,15-18,23,26-27,34-40,51,59H,9,14,19-22,24-25,49-50H2,1-3H3,(H,52,64)(H,53,61)(H,54,65)(H,55,62)(H,56,60)(H,57,63)(H,58,66)(H,67,68)/t27-,34+,35+,36+,37+,38+,39+,40+/m1/s1

Technical Data

Appearance: Solid Power

Purity: ≥98% (or refer to the Certificate of Analysis)

Shipping Condition: Shipped under ambient temperature as non-hazardous chemical or refer to Certificate of Analysis

Storage Condition: Dry, dark and -20 oC for 1 year or refer to the Certificate of Analysis.

Shelf Life: ≥12 months if stored properly.

Stock Solution Storage: 0 - 4 oC for 1 month or refer to the Certificate of Analysis.

Drug Formulation: To be determined

HS Tariff Code: 382200

Products are for research use only. Not for human use.

Payment & Security

PayPal Venmo

Your payment information is processed securely. We do not store credit card details nor have access to your credit card information.

You may also like

Recently viewed