Description
ZEN-3219 is a BET inhibitor with IC50s of 0.48, 0.16 and 0.47 μM for BRD4(BD1), BRD4(BD2) and BRD4(BD1BD2), respectively. ZEN-3219 can be used to form PROTACs to induce degradation of BRD4.
Product information
CAS Number: 1952264-34-4
Molecular Weight: 322.36
Formula: C19H18N2O3
Chemical Name: 5-(3,5-dimethyl-1,2-oxazol-4-yl)-1-{[4-(oxiran-2-yl)phenyl]methyl}-1,2-dihydropyridin-2-one
Smiles: CC1ON=C(C)C=1C1=CN(CC2C=CC(=CC=2)C2CO2)C(=O)C=C1
InChiKey: IELJHNIVCXDKQD-UHFFFAOYSA-N
InChi: InChI=1S/C19H18N2O3/c1-12-19(13(2)24-20-12)16-7-8-18(22)21(10-16)9-14-3-5-15(6-4-14)17-11-23-17/h3-8,10,17H,9,11H2,1-2H3
Technical Data
Appearance: Solid Power
Purity: ≥98% (or refer to the Certificate of Analysis)
Shipping Condition: Shipped under ambient temperature as non-hazardous chemical or refer to Certificate of Analysis
Storage Condition: Dry, dark and -20 oC for 1 year or refer to the Certificate of Analysis.
Shelf Life: ≥12 months if stored properly.
Stock Solution Storage: 0 - 4 oC for 1 month or refer to the Certificate of Analysis.
Drug Formulation: To be determined
HS Tariff Code: 382200
Products are for research use only. Not for human use.
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