MRS2179 tetrasodium - CAS# 1454889-37-2


Catalog No. Size PriceQuantity
M17422-C Contact sales@xcessbio.com for quotation $100

Description

MRS2179 tetrasodium is a competitive P2Y1 receptor antagonist, with a Kb of 102 nM and a pA2 of 6.99 for turkey P2Y1 receptor. MRS2179 tetrasodium is selective for P2Y1 over P2X1 (IC50=1.15 µM), P2X3 (12.9 µM), P2X2, P2X4, P2Y2, P2Y4, and P2Y6 receptors. MRS2179 tetrasodium inhibits platelet aggregation.

Product information

CAS Number: 1454889-37-2

Molecular Weight: 513.16

Formula: C11H13N5Na4O9P2

Chemical Name: tetrasodium (2R,3S,5S)-5-[6-(methylamino)-9H-purin-9-yl]-2-[(phosphonatooxy)methyl]oxolan-3-yl phosphate

Smiles: [Na+].[Na+].[Na+].[Na+].CNC1=NC=NC2=C1N=CN2[C@@H]1C[C@H](OP([O-])([O-])=O)[C@@H](COP([O-])([O-])=O)O1

InChiKey: XLPQPYQWGFCKEY-IDAKGYGSSA-J

InChi: InChI=1S/C11H17N5O9P2.4Na/c1-12-10-9-11(14-4-13-10)16(5-15-9)8-2-6(25-27(20,21)22)7(24-8)3-23-26(17,18)19;;;;/h4-8H,2-3H2,1H3,(H,12,13,14)(H2,17,18,19)(H2,20,21,22);;;;/q;4*+1/p-4/t6-,7+,8-;;;;/m0..../s1

Technical Data

Appearance: Solid Power

Purity: ≥98% (or refer to the Certificate of Analysis)

Shipping Condition: Shipped under ambient temperature as non-hazardous chemical or refer to Certificate of Analysis

Storage Condition: Dry, dark and -20 oC for 1 year or refer to the Certificate of Analysis.

Shelf Life: ≥12 months if stored properly.

Stock Solution Storage: 0 - 4 oC for 1 month or refer to the Certificate of Analysis.

Drug Formulation: To be determined

HS Tariff Code: 382200

How to use

In Vivo:

MRS2179 (50 mg/kg; i.p.) prolongs the bleeding time.

Products are for research use only. Not for human use.

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