LAS101057


Catalog No. Size PriceQuantity
M21808-C Contact sales@xcessbio.com for quotation $100Unavailable

Description

LAS101057 is a potent, selective, and orally efficacious A2B receptor antagonist.

Product information

CAS Number: 925676-48-8

Molecular Weight: 335.34

Formula: C18H14FN5O

Chemical Name: N-[5-(3-fluoropyridin-4-yl)-6-(pyridin-3-yl)pyrazin-2-yl]cyclopropanecarboxamide

Smiles: O=C(NC1=CN=C(C(=N1)C1C=NC=CC=1)C1=CC=NC=C1F)C1CC1

InChiKey: XUYURJQIMYCWBB-UHFFFAOYSA-N

InChi: InChI=1S/C18H14FN5O/c19-14-9-21-7-5-13(14)17-16(12-2-1-6-20-8-12)23-15(10-22-17)24-18(25)11-3-4-11/h1-2,5-11H,3-4H2,(H,23,24,25)

Technical Data

Appearance: Solid Power

Purity: ≥98% (or refer to the Certificate of Analysis)

Solubility: DMSO : ≥ 125 mg/mL (372.76 mM).

Shipping Condition: Shipped under ambient temperature as non-hazardous chemical or refer to Certificate of Analysis

Storage Condition: Dry, dark and -20 oC for 1 year or refer to the Certificate of Analysis.

Shelf Life: ≥12 months if stored properly.

Stock Solution Storage: 0 - 4 oC for 1 month or refer to the Certificate of Analysis.

Drug Formulation: To be determined

HS Tariff Code: 382200

How to use

In Vivo:

At 3 mg/kg, LAS101057 is active in preventing Acetyl-β-methylcholine-induced AHR, and at 10 mg/kg it inhibits AHR to Acetyl-β-methylcholine to a level virtually equal to that seen with Hexadecadrol at 1 mg/kg.

Products are for research use only. Not for human use.

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