Description
ZEN-3862 is a BET inhibitor with IC50s of 0.16 and 0.13 μM for BRD4(BD1) and BRD4(BD2) , respectively. ZEN-3862 can be used to form PROTACs to induce degradation of BRD4.
Product information
CAS Number: 1952264-33-3
Molecular Weight: 340.35
Formula: C19H17FN2O3
Chemical Name: 5-(3,5-dimethyl-1,2-oxazol-4-yl)-1-{[3-fluoro-4-(oxiran-2-yl)phenyl]methyl}-1,2-dihydropyridin-2-one
Smiles: CC1ON=C(C)C=1C1=CN(CC2C=C(F)C(=CC=2)C2CO2)C(=O)C=C1
InChiKey: VQHDSZCBMWYGEK-UHFFFAOYSA-N
InChi: InChI=1S/C19H17FN2O3/c1-11-19(12(2)25-21-11)14-4-6-18(23)22(9-14)8-13-3-5-15(16(20)7-13)17-10-24-17/h3-7,9,17H,8,10H2,1-2H3
Technical Data
Appearance: Solid Power
Purity: ≥98% (or refer to the Certificate of Analysis)
Shipping Condition: Shipped under ambient temperature as non-hazardous chemical or refer to Certificate of Analysis
Storage Condition: Dry, dark and -20 oC for 1 year or refer to the Certificate of Analysis.
Shelf Life: ≥12 months if stored properly.
Stock Solution Storage: 0 - 4 oC for 1 month or refer to the Certificate of Analysis.
Drug Formulation: To be determined
HS Tariff Code: 382200
Products are for research use only. Not for human use.
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