TRV130 Racemate


Catalog No. Size PriceQuantity
M8467-2 Solid 2 mg $130
M8467-10 Solid 10 mg $390

Description

TRV130 is a µ- opioid receptor agonist, that is currently under evaluation in human clinical trials for the treatment of acute severe pain. TRV130 is a functionally selective μ-opioid receptor agonist developed by Trevena Inc. TRV130 elicits robust G protein signaling, with potency and efficacy similar to morphine, but with far less β-arrestin 2 recruitment and receptor internalization, it displays less adverse effects than morphine. (http://en.wikipedia.org/wiki/TRV130). Oliceridine is now discontinued since it was recently listed as a controlled substance.

Product information

CAS Number: 1401028-25-8

Molecular Weight: 386.55

Formula: C22H30N2O2S

Synonym:

Oliceridine racemate

TRV-130 Racemate

Chemical Name: [(3-methoxythiophen-2-yl)methyl]({2-[9-(pyridin-2-yl)-6-oxaspiro[4.5]decan-9-yl]ethyl})amine

Smiles: COC1C=CSC=1CNCCC1(CCOC2(C1)CCCC2)C1=CC=CC=N1

InChiKey: DMNOVGJWPASQDL-UHFFFAOYSA-N

InChi: InChI=1S/C22H30N2O2S/c1-25-18-7-15-27-19(18)16-23-13-10-21(20-6-2-5-12-24-20)11-14-26-22(17-21)8-3-4-9-22/h2,5-7,12,15,23H,3-4,8-11,13-14,16-17H2,1H3

Technical Data

Appearance: Solid Power

Purity: ≥98% (or refer to the Certificate of Analysis)

Shipping Condition: Shipped under ambient temperature as non-hazardous chemical or refer to Certificate of Analysis

Storage Condition: Dry, dark and -20 oC for 1 year or refer to the Certificate of Analysis.

Shelf Life: ≥12 months if stored properly.

Stock Solution Storage: 0 - 4 oC for 1 month or refer to the Certificate of Analysis.

Drug Formulation: To be determined

HS Tariff Code: 382200

Products are for research use only. Not for human use.

Payment & Security

PayPal Venmo

Your payment information is processed securely. We do not store credit card details nor have access to your credit card information.

Estimate shipping

You may also like

Recently viewed